SCHEMBL22348708

SCHEMBL22348708

O=C(O)Nc1cccc(N(CC23CCC(c4noc(C5(F)CC5)n4)(CC2)CC3)C(=O)C2CC(O)(C(F)(F)F)C2)c1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.59
NR1I2 O75469 5/20 0.59
CYP2C9 P11712 5/20 0.59
CYP2C19 P33261 5/20 0.59
ABCB11 O95342 1/20 0.59
UGT1A1 P22309 1/20 0.59
FXR2 P51116 1/20 0.59
KCNH2 Q12809 1/20 0.59
SLCO1B3 Q9NPD5 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29458218 0.90 NR1H4 (0.57) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22348624 0.88 NR1H4 (0.60) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22347261 0.88 NR1H4 (0.62) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22347262 0.88 NR1H4 (0.62) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22348571 0.85 NR1H4 (0.53) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL25992771 0.81 NR1H4 (0.59) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22354218 0.80 NR1H4 (0.60) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22348707 0.78 NR1H4 (0.53) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22347534 0.76 NR1H4 (0.76) NR1H4NR1I2CYP2C9CYP2C19ABCB11
SCHEMBL22348448 0.76 NR1H4 (0.71) NR1H4NR1I2CYP2C9CYP2C19ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3924333-A1 SUBSTITUTED AMIDE COMPOUNDS USEFUL AS FARNESOID X RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2021-12-22 EP disclosed
WO-2020168149-A1 SUBSTITUTED AMIDE COMPOUNDS USEFUL AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed