SCHEMBL22352897

SCHEMBL22352897

O=C(C1CCC(F)(F)CC1)N(CCCCCc1noc(C(F)(F)F)n1)c1cccc(-c2cnc(C3CC3)nc2)c1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 16/20 0.48
NR1I2 O75469 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
HDAC1 Q13547 4/20 0.43
HDAC8 Q9BY41 4/20 0.43
HDAC6 Q9UBN7 4/20 0.43
HDAC5 Q9UQL6 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24451779 0.90 NR1H4 (0.46) NR1H4NR1I2CYP2C9CYP2C19HDAC1
SCHEMBL22352662 0.88 NR1H4 (0.48) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24452240 0.85 NR1H4 (0.58) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24452393 0.82 NR1H4 (0.51) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24452408 0.81 NR1H4 (0.43) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL22348191 0.81 NR1H4 (0.68) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24452480 0.81 NR1H4 (0.51) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24452395 0.81 NR1H4 (0.47) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24451786 0.81 NR1H4 (0.44) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24452472 0.80 NR1H4 (0.42) NR1H4NR1I2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020168148-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed