SCHEMBL22354080

SCHEMBL22354080

CCOc1ncc(-c2cccc(N(CC34CCC(c5ccc(C(F)(F)F)cn5)(CC3)CC4)C(=O)CCCF)c2)cn1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.65
NR1I2 O75469 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24259340 0.90 NR1H4 (0.63) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL22347348 0.86 NR1H4 (0.87) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL22354183 0.84 NR1H4 (0.56) NR1H4
SCHEMBL22354078 0.83 NR1H4 (0.69) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24259211 0.80 NR1H4 (0.75) NR1H4
SCHEMBL22347178 0.79 NR1H4 (1.00) NR1H4
SCHEMBL22353588 0.77 NR1H4 (1.00) NR1H4NR1I2CYP2C9CYP2C19
SCHEMBL24259233 0.77 NR1H4 (0.74) NR1H4
SCHEMBL22353590 0.77 NR1H4 (1.00) NR1H4
SCHEMBL25992661 0.76 NR1H4 (0.87) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020168143-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed