SCHEMBL22396409

SCHEMBL22396409

COc1cc(C(=N)NO)cnc1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
CA6 P23280 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
CA3 P07451 1/20 0.40
PKM P14618 1/20 0.40
CA5A P35218 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
TPMT P51580 2/20 0.39
PTGS2 P35354 1/20 0.38
P4HTM Q9NXG6 3/20 0.38
HPGDS O60760 1/20 0.37
HTT P42858 1/20 0.37
TSHR P16473 1/20 0.37
HDAC1 Q13547 5/20 0.36
HDAC6 Q9UBN7 5/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8768358 0.82 CA12 (0.53) CA12CA1CA2CA4CA6
SCHEMBL8787360 0.81 KDM4E (0.50) CA12CA1CA2CA4CA6
SCHEMBL8874902 0.75 CA12 (0.49) CA12CA1CA2CA4CA6
SCHEMBL3371450 0.74 LCK (0.44) CA12CA1CA2CA4CA6
SCHEMBL20943958 0.73 RECQL (0.44) CA12CA1CA2CA4CA6
SCHEMBL27393841 0.73 CYP2C9 (0.55) CA12CA1CA2CA7CA9
SCHEMBL20943959 0.73 RECQL (0.44) CA12CA1CA2CA4CA6
SCHEMBL22396419 0.73 LCK (0.41) CA12CA1CA2CA4CA6
SCHEMBL8786409 0.73 TP53 (0.55) L3MBTL1
Hydrochloric Acid SCHEMBL17161072 0.73 LCK (0.43) CA12CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704113-A1 BRIDGED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2020-09-09 EP disclosed