SCHEMBL22397989

SCHEMBL22397989

O=[N+]([O-])c1ccc(C=Cc2nc(COc3ccc(CCCCn4ccnn4)cc3)co2)c(F)c1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.62
MINK1 Q8N4C8 1/20 0.62
CA9 Q16790 2/20 0.33
CYP19A1 P11511 2/20 0.33
LMNA P02545 1/20 0.32
CNR1 P21554 2/20 0.32
ACHE P22303 2/20 0.32
CNR2 P34972 2/20 0.32
FFAR1 O14842 1/20 0.32
MAPT P10636 3/20 0.31
CA12 O43570 1/20 0.31
CA2 P00918 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22397986 1.00 ERBB2 (0.62) ERBB2MINK1CA9CYP19A1LMNA
SCHEMBL22397998 0.91 ERBB2 (0.59) ERBB2MINK1CA9CYP19A1LMNA
SCHEMBL28480665 0.91 ERBB2 (0.59) ERBB2MINK1CA9CYP19A1LMNA
SCHEMBL6582276 0.89 ERBB2 (0.68) ERBB2MINK1FFAR1MAPT
SCHEMBL6582279 0.89 ERBB2 (0.68) ERBB2MINK1FFAR1MAPT
SCHEMBL22398048 0.88 ERBB2 (0.47) ERBB2MINK1CA9CYP19A1LMNA
SCHEMBL28476214 0.88 ERBB2 (0.47) ERBB2MINK1CA9CYP19A1LMNA
SCHEMBL22398054 0.88 ERBB2 (0.47) ERBB2MINK1CA9CYP19A1LMNA
SCHEMBL22398043 0.88 ERBB2 (0.47) ERBB2MINK1CA9CYP19A1LMNA
SCHEMBL22397950 0.88 ERBB2 (0.74) ERBB2MINK1CYP19A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111886234-B Heterocyclic mitochondrial activity inhibitors and uses thereof 蒙特利尔大学 2023-12-15 CN disclosed
CN-111886234-A Heterocyclic mitochondrial activity inhibitors and uses thereof 蒙特利尔大学 2020-11-03 CN disclosed
EP-3704111-A1 HETEROCYCLIC MITOCHONDRIAL ACTIVITY INHIBITORS AND USES THEREOF Université de Montréal (CA) 2020-09-09 EP disclosed