SCHEMBL224067

SCHEMBL224067

O=C=Nc1cccc2cccc(N=C=O)c12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.60
ALDH1A1 P00352 6/20 0.41
HSD17B10 Q99714 5/20 0.41
HPGD P15428 4/20 0.41
TSHR P16473 4/20 0.41
CYP1A2 P05177 3/20 0.41
CYP1A1 P04798 2/20 0.41
CYP1B1 Q16678 2/20 0.41
GABRA1 P14867 1/20 0.40
GABRB2 P47870 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
ABCB11 O95342 1/20 0.39
NR3C1 P04150 1/20 0.39
ADRA2A P08913 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ALOX15 P16050 1/20 0.39
ADRA2C P18825 1/20 0.39
MAOA P21397 1/20 0.39
DRD1 P21728 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3669277 0.85 CYP3A4 (0.50) CYP3A4ALDH1A1HSD17B10HPGDTSHR
SCHEMBL11430534 0.84 CYP3A4 (0.46) CYP3A4ALDH1A1HSD17B10HPGDTSHR
Alpha-Naphthylisocyanate SCHEMBL29400034 0.79 CYP1A2 (0.64) CYP3A4ALDH1A1HSD17B10HPGDTSHR
Alpha-Naphthylisocyanate SCHEMBL374 0.79 CYP1A2 (0.64) CYP3A4ALDH1A1HSD17B10HPGDTSHR
SCHEMBL9229488 0.79 CYP3A4 (0.54) CYP3A4ALDH1A1HSD17B10HPGDTSHR
SCHEMBL9251624 0.79 CYP3A4 (0.54) CYP3A4ALDH1A1HSD17B10HPGDTSHR
SCHEMBL15431 0.78 CYP3A4 (0.64) CYP3A4ALDH1A1HSD17B10HPGDTSHR
SCHEMBL29395383 0.78 CYP3A4 (0.64) CYP3A4ALDH1A1HSD17B10HPGDTSHR
Alpha-Naphthylisocyanate SCHEMBL3333508 0.78 CYP1A2 (0.62) CYP3A4ALDH1A1HSD17B10HPGDTSHR
SCHEMBL29370250 0.77 CYP3A4 (0.62) CYP3A4ALDH1A1HSD17B10HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 759 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117820601-A Naphthalene diisocyanate composition, preparation method and application thereof 万华化学集团股份有限公司 2024-04-05 CN claimed
US-20240110002-A1 NOVEL POLYURETHANE OR POLYURETHANE-UREA COMPOSITION WITH ENHANCED LOW TEMPERATURE PERFORMANCE INGEVITY UK LTD (GB) 2024-04-04 US claimed
WO-2024068129-A1 NOVEL POLYURETHANE OR POLYURETHANE-UREA COMPOSITION WITH ENHANCED LOW TEMPERATURE PERFORMANCE INGEVITY UK LTD. (GB) 2024-04-04 WO claimed
CN-112384496-B Method for recovering diisocyanate from distillation residue 科思创德国股份有限公司 2024-02-02 CN claimed
CN-116178668-A Naphthalene diisocyanate composition and preparation method and application thereof 万华化学集团股份有限公司 2023-05-30 CN claimed
US-20230159693-A1 CURABLE COMPOSITIONS CONTAINING ISOCYANATE-BASED TOUGHENERS KANEKA AEROSPACE LLC (US) 2023-05-25 US claimed
US-20230050973-A1 METHOD FOR RECOVERING DIISOCYANATES FROM DISTILLATION RESIDUES COVESTRO DEUTSCHLAND AG (DE) 2023-02-16 US claimed
US-20210369911-A1 HYDROGEL COMPOSITIONS UNIVERSITÉ DE HAUTE-ALSACE (FR) 2021-12-02 US claimed
US-20210284603-A1 METHOD FOR EXTRACTING DIISOCYANATES FROM DISTILLATION RESIDUES COVESTRO DEUTSCHLAND AG (DE) 2021-09-16 US claimed
US-20210276944-A1 METHOD FOR RECOVERING DIISOCYANATES FROM DISTILLATION RESIDUES COVESTRO DEUTSCHLAND AG (DE) 2021-09-09 US claimed
WO-2003016247-A2 POLYMERIC URETHANE ESTER QUATS AND THEIR USE IN PERSONAL CARE COMPOSITIONS ALZO INTERNATIONAL, INC. (US) 2003-02-27 WO claimed
EP-0694532-B1 Perfluoroalkyl sulfide, sulfone, polysulfone and polysulfide diols CIBA SC HOLDING AG (CH) 2000-05-31 EP claimed
US-5998510-A POLYESTERURETHANE COPOLYMER PREMIX, INC. (US) 1999-12-07 US claimed
US-5708119-A POLYURETHANES FOR WATERPROOFING AND OIL REPELLENTS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-01-13 US claimed
US-5663273-A APPLYING TO IMPART OIL AND WATER REPELLENCY CIBA-GEIGY CORPORATION (US) 1997-09-02 US claimed
EP-0694532-A1 Perfluoroalkyl sulfide, sulfone, polysulfone and polysulfide diols CIBA-GEIGY AG (CH) 1996-01-31 EP claimed
EP-0690039-A2 Poly-perfluoroalkyl-substituted alcohols and acids, and derivatives thereof CIBA-GEIGY AG (CH) 1996-01-03 EP claimed
US-5200493-A Polyurethanes and polythiourethanes; protective coatings; oil repellents; waterproofing; antisoilants CIBA-GEIGY CORPORATION (US) 1993-04-06 US claimed
EP-0048117-A2 In-mold coating compositions containing a non-isocyanate-reactive unsaturated resin, a non-isocyanate-reactive monomer and a free isocyanate-containing compound ICI AMERICAS INC. (US) 1982-03-24 EP claimed
US-4105622-A PROCESS FOR THE PREPARATION OF FLAME RETARDANT THERMOPLASTIC RESIN COMPOSITIONS DAINIPPON INC. & CHEMICALS INC. (JP) 1978-08-08 US claimed