SCHEMBL22444686

SCHEMBL22444686

O=C(NC(CCc1ccc(C(F)(F)F)c(Cl)c1)C(=O)OCc1ccccc1)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
PTPN1 P18031 5/20 0.45
MDM2 Q00987 2/20 0.42
TNF P01375 1/20 0.41
IDO1 P14902 1/20 0.41
MDM4 O15151 2/20 0.40
TP53 P04637 2/20 0.40
EPHX2 P34913 1/20 0.39
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29634045 1.00 HDAC1 (0.46) HDAC1HDAC2PTPN1MDM2TNF
SCHEMBL29634006 0.91 PTPN1 (0.48) HDAC1HDAC2PTPN1MDM2IDO1
SCHEMBL22444643 0.91 MDM2 (0.49) MDM2TNFMDM4TP53
SCHEMBL22454854 0.91 MDM2 (0.49) MDM2TNFMDM4TP53
SCHEMBL29709620 0.91 MDM2 (0.49) MDM2TNFMDM4TP53
SCHEMBL31072743 0.91 MDM2 (0.49) MDM2TNFMDM4TP53
SCHEMBL22444602 0.88 PPARA (0.45) HDAC1HDAC2KMT2A
SCHEMBL28741600 0.88 MDM4 (0.41) PTPN1MDM2MDM4TP53
SCHEMBL29633743 0.88 MDM4 (0.41) PTPN1MDM2MDM4TP53
SCHEMBL29277322 0.84 MDM2 (0.49) MDM2TNFMDM4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113692401-A Process for producing aromatic amino acid derivative 中外制药株式会社 2021-11-23 CN disclosed
WO-2020189540-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE 中外製薬株式会社 2020-09-24 WO disclosed