SCHEMBL22452985

SCHEMBL22452985

O=C(O)c1cccc(Nc2cccc(Nc3ccc(C45CC6CC(CC(C6)C4)C5)cc3Cl)c2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 2/20 0.43
HIF1A Q16665 5/20 0.38
EPAS1 Q99814 3/20 0.38
ALDH1A1 P00352 2/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AURKA O14965 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
KMT2A Q03164 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
NPC1 O15118 1/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
EPHX2 P34913 2/20 0.34
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453312 0.95 SERPINE1 (0.43) SERPINE1HIF1AEPAS1ALDH1A1CA1
SCHEMBL22452779 0.91 SERPINE1 (0.39) SERPINE1SMN1; SMN2AURKAMEN1KMT2A
SCHEMBL22453603 0.86 HIF1A (0.43) SERPINE1HIF1AEPAS1ALDH1A1SMN1; SMN2
SCHEMBL22452975 0.85 AURKA (0.36) SERPINE1HIF1AALDH1A1CA1CA2
SCHEMBL22453039 0.84 CA1 (0.34) ALDH1A1CA1CA2SMN1; SMN2AURKA
SCHEMBL22452750 0.84 NPC1 (0.38) SERPINE1HIF1AEPAS1MEN1POLB
SCHEMBL22452560 0.82 SERPINE1 (0.40) SERPINE1HIF1AALDH1A1AURKAMEN1
SCHEMBL22453416 0.82 HIF1A (0.42) SERPINE1HIF1AEPAS1ALDH1A1SMN1; SMN2
SCHEMBL22452478 0.81 HIF1A (0.40) SERPINE1HIF1AEPAS1EPHX2
SCHEMBL22452684 0.80 HIF1A (0.52) SERPINE1HIF1AEPAS1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed