SCHEMBL22490660

SCHEMBL22490660

CCOC(=O)c1cc2c(s1)CCN(C(=O)CCCO)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.49
F2 P00734 1/20 0.43
TPSAB1 Q15661 1/20 0.43
TPSD1 Q9BZJ3 1/20 0.43
TPSG1 Q9NRR2 1/20 0.43
KDM1A O60341 5/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
POLB P06746 1/20 0.39
MCHR1 Q99705 1/20 0.39
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22490661 0.89 HDAC6 (0.49) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL19609145 0.87 HDAC6 (0.47) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL976216 0.86 HDAC6 (0.55) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL3441905 0.84 HDAC6 (0.54) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL7801200 0.83 HDAC6 (0.70) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL1174301 0.81 ADORA1 (0.57) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL3310243 0.79 KDM4E (0.48) HDAC6KDM4EALDH1A1HPGDTDP1
SCHEMBL11176901 0.79 KDM4E (0.48) HDAC6KDM4EALDH1A1HPGDTDP1
SCHEMBL19086215 0.79 HDAC6 (0.49) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL11179036 0.79 KDM4E (0.47) HDAC6KDM4EALDH1A1HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12479797-B2 Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors Jubilant Epicore LLC (US) 2025-11-25 US disclosed
EP-3455204-B1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS Jubilant Epicore LLC (US) 2025-10-29 EP disclosed
US-20220281815-A1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS Jubilant Epicore LLC 2022-09-08 US disclosed
US-11352322-B2 Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors Jubilant Epicore LLC (US) 2022-06-07 US disclosed
US-11352322-B2 Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors Jubilant Epicore LLC (US) 2022-06-07 US disclosed
US-20200308110-A1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS Jubilant Epicore LLC 2020-10-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200308110-A1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS HDAC1, HDAC11, HDAC2 HDAC6 8/4885F2 4767/4885TPSAB1 619/4885
US-11352322-B2 Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors HDAC1, HDAC11, HDAC2 HDAC6 8/4885F2 4767/4885TPSAB1 619/4885
US-12479797-B2 Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors HDAC1, HDAC11, HDAC2 HDAC6 7/4885F2 4823/4885TPSAB1 1243/4885
US-20220281815-A1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS HDAC1, HDAC11, HDAC2 HDAC6 7/4885F2 4823/4885TPSAB1 1243/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.