SCHEMBL22490868

SCHEMBL22490868

CC(C)(NC(=O)CCl)c1nc(NS(=O)(=O)C2CC2)sc1Cl

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTPS1 P17812 18/20 0.39
CTPS2 Q9NRF8 2/20 0.34
EPHX2 P34913 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22490800 0.89 CTPS1 (0.36) CTPS1CTPS2ALDH1A1
SCHEMBL22490846 0.80 CTPS1 (0.37) CTPS1CTPS2EPHX2NR1H4
SCHEMBL22869128 0.80 CTPS1 (0.38) CTPS1CTPS2EPHX2NR1H4
SCHEMBL22490823 0.79 CTPS1 (0.35) CTPS1CTPS2
SCHEMBL22869102 0.78 CTPS1 (0.37) CTPS1CTPS2
SCHEMBL22490769 0.77 CTPS1 (0.50) CTPS1CTPS2
SCHEMBL30455530 0.71 CTPS1 (0.55) CTPS1
SCHEMBL21381744 0.70 CTPS1 (0.57) CTPS1
SCHEMBL30415979 0.70 CTPS1 (0.57) CTPS1
SCHEMBL22490727 0.69 CTPS1 (0.38) CTPS1CTPS2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3717465-B1 COMPOUNDS STEP PHARMA S A S (FR) 2026-01-21 EP disclosed
US-20250263407-A1 Compounds STEP PHARMA S.A.S. (FR) 2025-08-21 US disclosed
US-12319680-B2 Compounds STEP PHARMA S.A.S. (FR) 2025-06-03 US disclosed
US-20230183229-A1 Compounds SYGNATURE DISCOVERY LIMITED (GB) 2023-06-15 US disclosed
US-20230183229-A1 Compounds SYGNATURE DISCOVERY LIMITED (GB) 2023-06-15 US disclosed
US-20230183229-A1 Compounds SYGNATURE DISCOVERY LIMITED (GB) 2023-06-15 US disclosed
US-11505547-B2 Compounds STEP PHARMA S.A.S. (FR) 2022-11-22 US disclosed
US-20210380575-A1 COMPOUNDS SYGNATURE DISCOVERY LIMITED (GB) 2021-12-09 US disclosed
EP-3717465-A1 COMPOUNDS Step Pharma S.A.S. (FR) 2020-10-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230183229-A1 Compounds UGT1A1, CYP1A1, CYP1B1 CTPS1 2556/4885CTPS2 2833/4885EPHX2 1110/4885
US-12319680-B2 Compounds UGT1A1, CYP1A1, CYP1B1 CTPS1 2556/4885CTPS2 2833/4885EPHX2 1110/4885
US-20250263407-A1 Compounds CYP1A1, UGT1A1, CYP1A2 CTPS1 2586/4885CTPS2 2637/4885EPHX2 1004/4885
US-11505547-B2 Compounds UGT1A1, CYP1A1, CYP1B1 CTPS1 2556/4885CTPS2 2833/4885EPHX2 1110/4885
US-20210380575-A1 COMPOUNDS UGT1A1, CYP1A1, CYP1B1 CTPS1 2556/4885CTPS2 2833/4885EPHX2 1110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.