SCHEMBL22497746

SCHEMBL22497746

COc1cc2c(Oc3ccc(N(C(=O)C4(C(N)=O)CC4)c4ccc(F)cc4)cc3F)ccnc2cc1OCCCCCNC(=O)CS

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 2/20 0.56
HDAC8 Q9BY41 2/20 0.56
HDAC6 Q9UBN7 2/20 0.56
HDAC10 Q969S8 1/20 0.56
HDAC11 Q96DB2 1/20 0.56
MET P08581 16/20 0.54
AXL P30530 7/20 0.54
KDR P35968 4/20 0.54
RET P07949 3/20 0.54
KIT P10721 3/20 0.54
FLT3 P36888 3/20 0.54
PDGFRB P09619 2/20 0.54
MERTK Q12866 3/20 0.49
AURKA O14965 2/20 0.49
RIPK2 O43353 2/20 0.49
ABL1 P00519 2/20 0.49
EGFR P00533 2/20 0.49
ERBB2 P04626 2/20 0.49
NTRK1 P04629 2/20 0.49
LCK P06239 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28692805 0.92 HDAC2 (0.56) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL30786374 0.92 HDAC2 (0.56) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL29182979 0.92 HDAC2 (0.56) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL28686931 0.90 HDAC2 (0.57) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL15917325 0.89 HDAC2 (0.70) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL15918114 0.89 HDAC2 (0.70) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL15917470 0.89 HDAC2 (0.70) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL15917808 0.89 HDAC2 (0.70) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL15917659 0.89 HDAC2 (0.69) HDAC2HDAC8HDAC6HDAC10HDAC11
SCHEMBL15918162 0.89 HDAC2 (0.69) HDAC2HDAC8HDAC6HDAC10HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113924288-B Quinolinyl-containing compound, pharmaceutical composition and application thereof 北京普祺医药科技股份有限公司 2024-04-05 CN disclosed
CN-113924288-A Quinolyl-containing compound, pharmaceutical composition and application thereof 北京普祺医药科技有限公司 2022-01-11 CN disclosed
WO-2020200160-A1 QUINOLYL-CONTAINING COMPOUND AND PHARMACEUTICAL COMPOSITION, AND USE THEREOF 北京国鸿生物医药科技有限公司 2020-10-08 WO disclosed