SCHEMBL22497749

SCHEMBL22497749

C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OCC)cc1N(C)CCNC

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.88
IGF1R P08069 1/20 0.88
MLNR O43193 1/20 0.77
KDM1A O60341 1/20 0.77
ABCB11 O95342 1/20 0.77
ERBB2 P04626 1/20 0.77
INSR P06213 1/20 0.77
CHRM2 P08172 1/20 0.77
HTR1A P08908 1/20 0.77
ADORA3 P0DMS8 1/20 0.77
DRD2 P14416 1/20 0.77
NQO2 P16083 1/20 0.77
ADRA2C P18825 1/20 0.77
DRD1 P21728 1/20 0.77
ERBB3 P21860 1/20 0.77
SLC6A2 P23975 1/20 0.77
HTR2A P28223 1/20 0.77
HTR2C P28335 1/20 0.77
ADORA2A P29274 1/20 0.77
SLC6A4 P31645 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29860673 0.94 EGFR (1.00) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL30379658 0.94 EGFR (1.00) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL14661086 0.94 EGFR (1.00) EGFRIGF1RMLNRKDM1AABCB11
Hydrochloric Acid SCHEMBL30735819 0.93 EGFR (0.99) EGFRIGF1RMLNRKDM1AABCB11
Hydrochloric Acid SCHEMBL30735856 0.93 EGFR (0.99) EGFRIGF1RMLNRKDM1AABCB11
Hydrochloric Acid SCHEMBL26637892 0.93 EGFR (0.99) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL22509190 0.93 EGFR (0.88) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL22509155 0.91 EGFR (0.77) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL22509192 0.91 EGFR (0.85) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL30682157 0.91 EGFR (0.95) EGFRIGF1RMLNRKDM1AABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12258344-B2 Azaaromatic amide derivatives for the treatment of cancer SHENZHEN FORWARD PHARMACEUTICALS CO., LTD. (CN) 2025-03-25 US disclosed
US-20220177473-A1 AZAAROMATIC AMIDE DERIVATIVES FOR THE TREATMENT OF CANCER SHENZHEN FORWARD PHARMACEUTICALS CO., LTD. (CN) 2022-06-09 US disclosed
US-20220177473-A1 AZAAROMATIC AMIDE DERIVATIVES FOR THE TREATMENT OF CANCER SHENZHEN FORWARD PHARMACEUTICALS CO., LTD. (CN) 2022-06-09 US disclosed
EP-3950686-A1 N-HETEROAROMATIC AMIDE DERIVATIVES FOR TREATMENT OF CANCER Shenzhen Forward Pharmaceuticals Co., Ltd. (CN) 2022-02-09 EP disclosed
CN-113727982-A Azaaromatic cyclic amide derivatives for the treatment of cancer 深圳福沃药业有限公司 2021-11-30 CN disclosed
CN-111747931-A Azaaromatic cyclic amide derivatives for the treatment of cancer 深圳福沃药业有限公司 2020-10-09 CN disclosed
WO-2020200158-A1 N-HETEROAROMATIC AMIDE DERIVATIVES FOR TREATMENT OF CANCER 深圳福沃药业有限公司 2020-10-08 WO disclosed
WO-2020200158-A1 N-HETEROAROMATIC AMIDE DERIVATIVES FOR TREATMENT OF CANCER 深圳福沃药业有限公司 2020-10-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220177473-A1 AZAAROMATIC AMIDE DERIVATIVES FOR THE TREATMENT OF CANCER ERBB4, EGFR, ERBB2 EGFR 2/4885IGF1R 47/4885MLNR 487/4885
US-12258344-B2 Azaaromatic amide derivatives for the treatment of cancer ERBB4, EGFR, ERBB2 EGFR 2/4885IGF1R 47/4885MLNR 487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.