SCHEMBL2250264

SCHEMBL2250264

CC(C)C[C@H](N)C(=O)Nc1ccc2ncnc(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2c1

nearest known ligand 0.75

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 17/20 0.75
EGFR P00533 14/20 0.75
LCK P06239 1/20 0.75
KCNH2 Q12809 3/20 0.59
AURKA O14965 1/20 0.58
RPS6KB1 P23443 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28768471 0.91 ERBB2 (0.77) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL2322666 0.91 ERBB2 (0.77) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL2250011 0.86 EGFR (0.68) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL2249176 0.84 ERBB2 (0.79) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL2251397 0.83 ERBB2 (0.79) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL2251452 0.83 EGFR (0.70) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL27718944 0.83 EGFR (0.70) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL19479997 0.82 ERBB2 (0.77) ERBB2EGFRLCKKCNH2AURKA
SCHEMBL7236445 0.82 EGFR (0.81) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL2249350 0.81 EGFR (0.64) ERBB2EGFRLCKAURKARPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003658-B2 Quinazoline derivatives for inhibiting cancer cell growth and method for the preparation thereof HANMI HOLDINGS CO., LTD. (KR) 2011-08-23 US disclosed