Pf-06842874

Pf-06842874

SCHEMBL22553485

CC(=O)c1c(C)c2cnc(N[C@H]3CCOC[C@@H]3O)cc2n(C2CCCC2)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 1.00
CCND1 P24385 20/20 1.00
CCND3 P30281 20/20 1.00
CDK6 Q00534 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pf-06842874 SCHEMBL22553475 1.00 CDK4 (1.00) CDK4CCND1CCND3CDK6
Pf-06842874 SCHEMBL22553598 1.00 CDK4 (1.00) CDK4CCND1CCND3CDK6
Pf-06842874 SCHEMBL22553637 1.00 CDK4 (1.00) CDK4CCND1CCND3CDK6
Pf-06842874 SCHEMBL22553605 1.00 CDK4 (1.00) CDK4CCND1CCND3CDK6
SCHEMBL22553586 0.94 CDK4 (1.00) CDK4CCND1CCND3CDK6
SCHEMBL22553599 0.91 CDK4 (1.00) CDK4CCND1CCND3CDK6
SCHEMBL22553493 0.91 CDK4 (1.00) CDK4CCND1CCND3CDK6
SCHEMBL22553639 0.91 CDK4 (1.00) CDK4CCND1CCND3CDK6
SCHEMBL22566627 0.91 CDK4 (1.00) CDK4CCND1CCND3CDK6
SCHEMBL22553524 0.91 CDK4 (1.00) CDK4CCND1CCND3CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007697-A Antiproliferative agents for the treatment of PAH 辉瑞公司 2022-02-01 CN disclosed
US-11203594-B2 Anti-proliferative agents for treating PAH PFIZER INC. (US) 2021-12-21 US disclosed
US-20200331909-A1 ANTI-PROLIFERATIVE AGENTS FOR TREATING PAH PFIZER INC. (US) 2020-10-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11203594-B2 Anti-proliferative agents for treating PAH EDNRB, EDNRA, PAH CDK4 219/4885CCND1 108/4885CCND3 143/4885
US-20200331909-A1 ANTI-PROLIFERATIVE AGENTS FOR TREATING PAH EDNRB, EDNRA, PAH CDK4 219/4885CCND1 108/4885CCND3 143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.