SCHEMBL22604241

SCHEMBL22604241

CCCC(CC)c1c(Cl)cc(C(F)(F)F)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GABRA2 P47869 9/20 0.39
GABRB2 P47870 9/20 0.39
GABRB3 P28472 12/20 0.38
PDE2A O00408 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26462712 0.85 AR (0.37) GABRA2GABRB2GABRB3
SCHEMBL18896300 0.83 CYP3A4 (0.51)
SCHEMBL21725448 0.80 PDE2A (0.55) PDE2A
SCHEMBL22222362 0.78 KMT2A (0.36) PDE2A
SCHEMBL21164525 0.78 KMT2A (0.36) PDE2A
SCHEMBL18638714 0.76 PDE2A (0.44) GABRA2GABRB2GABRB3PDE2A
SCHEMBL22222395 0.72 PDE2A (0.34) PDE2A
SCHEMBL22898345 0.72 PDE2A (0.39) GABRA2GABRB2GABRB3PDE2A
SCHEMBL21725447 0.71 PDE2A (0.62) PDE2A
SCHEMBL19003603 0.70 PDE2A (0.43) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11331320-B2 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors INCYTE HOLDINGS CORPORATION (US) 2022-05-17 US disclosed
US-20200338077-A1 HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS INCYTE CORPORATION 2020-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200338077-A1 HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS JAK3, JAK1, JAK2 GABRA2 1824/4885GABRB2 1606/4885GABRB3 1423/4885
US-11331320-B2 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors JAK3, JAK1, JAK2 GABRA2 1824/4885GABRB2 1606/4885GABRB3 1423/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.