SCHEMBL2260665

SCHEMBL2260665

CCCC1CCCCC1C#N

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA4 P22748 1/20 0.48
ADRA2A P08913 2/20 0.33
ADRA2B P18089 2/20 0.33
ADRA2C P18825 2/20 0.33
ADRA1A P35348 1/20 0.33
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14620937 0.96 CA1 (0.43) CA1CA2CA4
SCHEMBL28886067 0.86 CYP1A2 (0.38) CA1CA2CA4CYP1A2
SCHEMBL2288404 0.82 CA1 (0.32) CA1CA2CA4
SCHEMBL19592339 0.82 CA1 (0.32) CA1CA2CA4
SCHEMBL2263208 0.82 EPHX1 (0.34) CA1CA2CA4CYP1A2
SCHEMBL2261801 0.80 EPHX1 (0.37) CA1CA2CA4CYP1A2
SCHEMBL20380947 0.80 CA1 (0.31) CA1CA2CA4
SCHEMBL24929562 0.77
SCHEMBL24929113 0.77
SCHEMBL24404223 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9814722-B2 Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors INCYTE HOLDINGS CORPORATION (US) 2017-11-14 US disclosed
EP-2217563-B1 Alpha-substituted cyclopentanecarbonitriles or cyclohexanecarbonitriles and their use in perfumery FIRMENICH & CIE (CH) 2013-01-30 EP disclosed
US-8003084-B2 α-substituted cyclopentanecarbonitriles or cyclohexanecarbonitriles and their use in perfumery FIRMENICH SA (CH) 2011-08-23 US disclosed
US-20100247467-A1 ALPHA-SUBSTITUTED CYCLOPENTANECARBONITRILES OR CYCLOHEXANECARBONITRILES AND THEIR USE IN PERFUMERY FIRMENICH SA (CH) 2010-09-30 US disclosed
EP-2217563-A2 ALPHA-SUBSTITUTED CYCLOPENTANECARBONITRILES OR CYCLOHEXANECARBONITRILES AND THEIR USE IN PERFUMERY Firmenich S.A. (CH) 2010-08-18 EP disclosed
WO-2009060378-A2 ALPHA-SUBSTITUTED CYCLOPENTANECARBONITRILES OR CYCLOHEXANECARBONITRILES AND THEIR USE IN PERFUMERY FIRMENICH SA (CH) 2009-05-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100247467-A1 ALPHA-SUBSTITUTED CYCLOPENTANECARBONITRILES OR CYCLOHEXANECARBONITRILES AND THEIR USE IN PERFUMERY PNN, FASN, CYP8B1 CA1 2439/4885CA2 2591/4885CA4 1865/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.