SCHEMBL22639708

SCHEMBL22639708

O=C(O)C1CCN(Cc2nc3ccccc3[nH]2)CC1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.66
GRIN2B Q13224 1/20 0.66
HTT P42858 1/20 0.63
DRD4 P21917 11/20 0.61
HPGD P15428 1/20 0.60
DRD2 P14416 2/20 0.57
NPC1 O15118 1/20 0.56
GAA P10253 1/20 0.56
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
CACNA1G O43497 1/20 0.53
CHRNA7 P36544 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15550981 0.89 HTT (0.61) GRIN1GRIN2BHTTDRD4HPGD
SCHEMBL5157052 0.82 HTT (0.84) GRIN1GRIN2BHTTDRD4HPGD
SCHEMBL16795300 0.82 DRD4 (0.67) GRIN1GRIN2BHTTDRD4HPGD
SCHEMBL4791717 0.82 CHRNA7 (0.77) GRIN1GRIN2BHTTDRD4HPGD
SCHEMBL6941438 0.81 HTT (0.69) GRIN1GRIN2BHTTDRD4HPGD
SCHEMBL7085421 0.80 IDO1 (0.67) GRIN1GRIN2BNPC1GAAKDM4E
SCHEMBL14338810 0.80 HPGD (0.55) GRIN1GRIN2BHTTDRD4HPGD
SCHEMBL7085424 0.80 IDO1 (0.67) GRIN1GRIN2BNPC1GAAKDM4E
SCHEMBL7086561 0.80 IDO1 (0.67) GRIN1GRIN2BNPC1GAAKDM4E
SCHEMBL1388535 0.80 GRIN2B (1.00) GRIN1GRIN2BHTTDRD4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10828281-B2 Non-hydrophobic compounds for use in treating metastasis and/or cartilage defect Friedrich-Alexander-Universität Erlangen-Nürnberg (DE) 2020-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10828281-B2 Non-hydrophobic compounds for use in treating metastasis and/or cartilage defect VIM, MATR3, TP53 GRIN1 4074/4885GRIN2B 4318/4885HTT 488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.