SCHEMBL22643135

SCHEMBL22643135

Cc1ccc(-c2cnn(CC(C)C)c2)cc1F

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 18/20 0.58
PRMT5 O14744 1/20 0.48
WDR77 Q9BQA1 1/20 0.48
GRIN2B Q13224 4/20 0.46
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19998601 0.84 KCNH2 (0.62) KCNH2PRMT5WDR77GRIN2B
SCHEMBL22642969 0.81 KCNH2 (0.63) KCNH2PRMT5WDR77GRIN2B
SCHEMBL16911740 0.80 PRMT5 (0.48) KCNH2PRMT5WDR77ACHE
SCHEMBL17130593 0.80 PRMT5 (0.48) KCNH2PRMT5WDR77ACHE
SCHEMBL16812740 0.80 KCNH2 (0.46) KCNH2PRMT5WDR77GRIN2B
SCHEMBL10094700 0.79 PDK2 (0.45) PRMT5WDR77ACHE
Hydrochloric Acid SCHEMBL16648539 0.79 KCNH2 (0.46) KCNH2PRMT5WDR77GRIN2B
SCHEMBL17795050 0.79 NAMPT (0.48) KCNH2PRMT5WDR77GRIN2BACHE
SCHEMBL16911242 0.78 PRMT5 (0.46) KCNH2PRMT5WDR77GRIN2BACHE
SCHEMBL19998585 0.78 KCNH2 (0.59) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970283-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-11-11 EP disclosed