SCHEMBL22650627

SCHEMBL22650627

CC(C)n1cnc2c(F)nc(-c3ccnc(Nc4ccc(N5CCCC(N(C)C)C5=O)cn4)n3)cc21

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.39
CDK6 Q00534 12/20 0.39
CCND3 P30281 11/20 0.39
CCND1 P24385 13/20 0.39
CCNA2 P20248 11/20 0.39
CDK2 P24941 10/20 0.39
CCNA1 P78396 3/20 0.39
GSK3B P49841 1/20 0.38
CDK1 P06493 9/20 0.36
CCNB1 P14635 8/20 0.36
CCNT1 O60563 5/20 0.35
CDK9 P50750 5/20 0.35
CDK7 P50613 5/20 0.35
CCNH P51946 5/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650536 0.91 JAK2 (0.34) CCNA2CDK2CCNA1CDK1CCNB1
SCHEMBL22650531 0.89 CDK6 (0.42) CDK4CDK6CCND3CCND1CCNA2
SCHEMBL22650619 0.89 CDK4 (0.40) CDK4CDK6CCND3CCND1CCNA2
SCHEMBL29491142 0.88 CDK4 (0.44) CDK4CDK6CCND3CCND1CCNA2
SCHEMBL22650933 0.88 CDK4 (0.44) CDK4CDK6CCND3CCND1CCNA2
SCHEMBL22650935 0.88 CDK4 (0.44) CDK4CDK6CCND3CCND1CCNA2
SCHEMBL22635855 0.88 CDK4 (0.44) CDK4CDK6CCND3CCND1CCNA2
SCHEMBL22650578 0.86 IKBKB (0.35) CCNA2CDK2CCNA1CDK1CCNB1
SCHEMBL22650574 0.86 CDK4 (0.43) CDK4CDK6CCND3CCND1CCNA2
SCHEMBL22650778 0.85 CDK4 (0.42) CDK4CDK6CCND3CCND1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed