SCHEMBL22650795

SCHEMBL22650795

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCCC(N(C)C)C5=O)cn4)n3)cc12

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 18/20 0.41
CCND1 P24385 9/20 0.41
CDK6 Q00534 9/20 0.41
CDK1 P06493 5/20 0.41
CCNB1 P14635 4/20 0.41
CCNA2 P20248 7/20 0.40
CDK2 P24941 6/20 0.40
CCNA1 P78396 3/20 0.40
GSK3B P49841 1/20 0.40
CCND3 P30281 6/20 0.40
CCNT1 O60563 2/20 0.37
CDK9 P50750 2/20 0.37
CDK7 P50613 1/20 0.37
CCNH P51946 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650419 0.91 JAK2 (0.38) CDK4CCND1CDK1CCNB1CDK9
SCHEMBL22650450 0.89 CDK4 (0.41) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650847 0.87 JAK2 (0.39) CDK4CCND1CDK1CCNB1CCNA2
SCHEMBL22650823 0.85 CDK4 (0.45) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650901 0.85 CDK4 (0.45) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650366 0.85 CDK4 (0.47) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650797 0.84 CDK4 (0.42) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL29491159 0.83 CDK4 (0.58) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22635854 0.83 CDK4 (0.58) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650924 0.83 CDK4 (0.48) CDK4CCND1CDK6CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed