SCHEMBL22650798

SCHEMBL22650798

CC(C)c1cnn2ccc(-c3nc(Nc4ccc(N5CCC(N6CC(F)(F)C6)CC5=O)cn4)ncc3F)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 19/20 0.42
CDK4 P11802 15/20 0.42
CCND1 P24385 7/20 0.40
CCNA2 P20248 7/20 0.40
CCND3 P30281 7/20 0.40
CDK2 P24941 4/20 0.40
CDK9 P50750 4/20 0.40
CCNT1 O60563 3/20 0.40
CDK7 P50613 1/20 0.40
CCNH P51946 1/20 0.40
MNAT1 P51948 1/20 0.40
CDK1 P06493 5/20 0.40
CYP2C9 P11712 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNE1 P24864 1/20 0.40
CYP2C19 P33261 1/20 0.40
CDK5 Q00535 1/20 0.40
KCNH2 Q12809 1/20 0.40
CDK5R1 Q15078 1/20 0.40
CCNK O75909 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650799 0.88 CDK6 (0.43) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650479 0.88 CDK6 (0.47) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650845 0.86 CDK6 (0.48) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650926 0.85 CDK4 (0.48) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650591 0.84 CDK6 (0.48) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650758 0.83 CDK4 (0.52) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650462 0.83 CDK6 (0.46) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650601 0.83 CDK6 (0.48) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650945 0.83 CDK6 (0.60) CDK6CDK4CCND1CCNA2CCND3
SCHEMBL22650486 0.82 CDK6 (0.54) CDK6CDK4CCND1CCNA2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed