SCHEMBL22650857

SCHEMBL22650857

COc1nc(-c2ccnc(Nc3ccc(CN4CCC(F)(F)C4)cn3)n2)cc2c1ncn2C(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 16/20 0.45
CCND1 P24385 14/20 0.45
CDK4 P11802 11/20 0.44
CDK1 P06493 5/20 0.44
CCNB1 P14635 2/20 0.44
CCND3 P30281 5/20 0.41
CDK2 P24941 5/20 0.38
CCNA2 P20248 4/20 0.38
CCNA1 P78396 2/20 0.38
DYRK2 Q92630 2/20 0.38
CCNT1 O60563 2/20 0.38
CDK7 P50613 2/20 0.38
CDK9 P50750 2/20 0.38
CCNH P51946 2/20 0.38
CIT O14578 1/20 0.37
GAK O14976 1/20 0.37
DYRK3 O43781 1/20 0.37
STK16 O75716 1/20 0.37
CCNK O75909 1/20 0.37
STK10 O94804 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650734 0.88 CDK6 (0.48) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650946 0.87 CDK6 (0.44) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650856 0.85 CDK6 (0.47) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650860 0.83 CDK6 (0.44) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650548 0.78 CDK4 (0.41) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650956 0.78 CDK6 (0.59) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650859 0.78 CDK4 (0.51) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650958 0.77 CDK4 (0.42) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650429 0.76 CCND1 (0.40) CDK6CCND1CDK4CDK1CCNB1
SCHEMBL22650513 0.75 CDK4 (0.36) CDK6CCND1CDK4CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed