SCHEMBL22650952

SCHEMBL22650952

COc1nc(-c2nc(Nc3ccc(N4CCN(CCS(C)(=O)=O)CC4=O)cn3)ncc2F)cc2c1nc(C)n2C(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 18/20 0.49
CDK6 Q00534 17/20 0.49
CDK2 P24941 16/20 0.49
CCNA2 P20248 4/20 0.49
CCND3 P30281 4/20 0.49
CDK1 P06493 9/20 0.47
CDK7 P50613 7/20 0.47
CDK9 P50750 7/20 0.47
CDK5 Q00535 3/20 0.47
CCNB1 P14635 6/20 0.46
CCNE1 P24864 6/20 0.46
EGFR P00533 3/20 0.46
CCNT1 O60563 2/20 0.46
NTRK1 P04629 2/20 0.46
BRAF P15056 2/20 0.46
KDR P35968 2/20 0.46
MAPK8 P45983 2/20 0.46
CCNH P51946 2/20 0.46
MNAT1 P51948 2/20 0.46
MAPK10 P53779 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650452 0.92 CDK4 (0.54) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650557 0.90 CDK4 (0.53) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650525 0.90 CDK4 (0.47) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650528 0.87 CDK4 (0.45) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650735 0.85 CDK4 (0.48) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650613 0.85 CDK4 (0.48) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650632 0.84 CDK6 (0.46) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650543 0.84 CDK4 (0.44) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650954 0.83 CDK6 (0.50) CDK4CDK6CDK2CCNA2CCND3
SCHEMBL22650458 0.83 CDK6 (0.55) CDK4CDK6CDK2CCNA2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed