SCHEMBL22666348

SCHEMBL22666348

Cc1ncc(OCC2C[C@H]2C(=O)Nc2ccc(F)cn2)c(C)n1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.62
HCRTR2 O43614 20/20 0.62
KCNH2 Q12809 6/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22729371 1.00 HCRTR1 (0.62) HCRTR1HCRTR2KCNH2
SCHEMBL20859727 1.00 HCRTR1 (0.62) HCRTR1HCRTR2KCNH2
SCHEMBL2116797 0.77 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
SCHEMBL2118675 0.77 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
SCHEMBL22666162 0.76 FFAR4 (0.43) HCRTR1HCRTR2KCNH2
SCHEMBL10266354 0.76 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
SCHEMBL2610611 0.76 HCRTR1 (0.87) HCRTR1HCRTR2KCNH2
SCHEMBL16638939 0.76 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
SCHEMBL22729373 0.75 GRM5 (0.39) HCRTR1HCRTR2KCNH2
SCHEMBL2610676 0.75 HCRTR1 (0.69) HCRTR1HCRTR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021145373-A1 DRUG SUBSTANCE OF LEMBOREXANT AND MEDICINAL COMPOSITION COMPRISING SAME エーザイ・アール・アンド・ディー・マネジメント株式会社 2021-07-22 WO disclosed
WO-2020230800-A1 METHOD AND COMPOUND USEFUL IN PREPARATION OF OREXIN-2 RECEPTOR ANTAGONIST, AND LEMBOREXANT HAVING FEW IMPURITIES エーザイ・アール・アンド・ディー・マネジメント株式会社 2020-11-19 WO disclosed