SCHEMBL226964

SCHEMBL226964

[NH]C(=O)CBr

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2300400 0.72
Bromoacetic Acid SCHEMBL1332313 0.67
SCHEMBL5106 0.67
SCHEMBL180158 0.67
Bromoacetic Acid SCHEMBL7617676 0.67
SCHEMBL5518651 0.67
Bromoacetic Acid SCHEMBL1332022 0.67
Bromoacetic Acid SCHEMBL1332132 0.67
SCHEMBL34263 0.67
Bromoacetic Acid SCHEMBL16011275 0.67 TSHR (1.00)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1455 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023198195-A1 CONJUGATE COMPRISING TOLL-LIKE RECEPTOR AGONIST MABSOFT THERAPEUTICS (SHANGHAI) CO., LTD. (CN) 2023-10-19 WO claimed
EP-3318555-B1 BIFUNCTIONAL CHELATING AGENTS BWXT MEDICAL LTD (CA) 2023-08-16 EP claimed
EP-4073204-B1 LUMINESCENT LANTHANIDE(III) CHELATES UNIOGEN OY (FI) 2023-08-09 EP claimed
CN-115671274-A Method for linking carrier protein and polysaccharide into conjugate by covalent bond and application 普大生物科技(泰州)有限公司 2023-02-03 CN claimed
US-20230025102-A1 LUMINESCENT LANTHANIDE(III) CHELATES UNIOGEN OY (FI) 2023-01-26 US claimed
WO-2022264970-A1 MITOCHONDRIA-SELECTIVE NITROXYL RADICAL COMPOUND 国立大学法人東海国立大学機構 2022-12-22 WO claimed
WO-2022264971-A1 METHOD FOR EVALUATING QUALITY OF SPERM 国立大学法人東海国立大学機構 2022-12-22 WO claimed
US-20220280530-A1 PREVENTION OR TREATMENT OF DISEASES AND DISORDERS ASSOCIATED WITH TISSUE DAMAGE Anhui Newstar Pharmaceutical Development Co., Ltd. (CN) 2022-09-08 US claimed
CN-114728009-A Preventing or treating diseases and disorders associated with tissue damage 李晓祥 2022-07-08 CN claimed
EP-3990446-A1 NOVEL LUMINESCENT LANTHANIDE CHELATE REPORTERS, BIOSPECIFIC BINDING REACTANTS LABELLED WITH NOVEL LUMINESCENT LANTHANIDE CHELATE REPORTERS AND THEIR USE Radiometer Turku Oy (FI) 2022-05-04 EP claimed
EP-0367223-A2 Chelants possessing ortho ligating functionality and complexes thereof THE DOW CHEMICAL COMPANY (US) 1990-05-09 EP claimed
EP-0353450-A1 Macrocyclic bifunctional chelants, complexes thereof and their antibody conjugates THE DOW CHEMICAL COMPANY (US) 1990-02-07 EP claimed
WO-1989012631-A1 MACROCYCLIC BIFUNCTIONAL CHELANTS, COMPLEXES THEREOF AND THEIR ANTIBODY CONJUGATES THE DOW CHEMICAL COMPANY (US) 1989-12-28 WO claimed
US-4751288-A COLORFASTNESS BASF AKTIENGESELLSCHAFT (DE) 1988-06-14 US claimed
EP-0034759-B1 CHROMOGEN CEPHALOSPORINS AND PROCESS FOR THEIR PREPARATION HOECHST AKTIENGESELLSCHAFT (DE) 1986-01-02 EP claimed
EP-0044134-B1 COMPOSITION FOR REDUCING INTRAOCULAR PRESSURE UNIVERSITY OF FLORIDA (US) 1985-06-05 EP claimed
US-4448880-A Detection of β-lactamase utilizing a chromophoric cephalosporin composition HOECHST AG. (DE) 1984-05-15 US claimed
US-4407815-A AMINO ACID DERIVATIVE ANTIBIOTICS BEECHAM GROUP LIMITED (GB) 1983-10-04 US claimed
EP-0018001-B1 CHROMOPHORIC CEPHALOSPORIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR UTILISATION, COMPOSITIONS CONTAINING THEM AND THEIR PREPARATION HOECHST AKTIENGESELLSCHAFT (DE) 1983-05-25 EP claimed
US-4353824-A DETECTORS OF BETA-LACTAMASES HOECHST AKTIENGESELLSCHAFT (DE) 1982-10-12 US claimed