SCHEMBL2269788

SCHEMBL2269788

Cc1c(Cc2cccc(S(=O)(=O)c3ccc(Cl)cc3)c2)c2cc(F)ccc2n1CC(=O)O

nearest known ligand 0.68

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 20/20 0.68
AKR1B1 P15121 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2269355 0.93 PTGDR2 (0.72) PTGDR2
SCHEMBL2272823 0.92 PTGDR2 (0.78) PTGDR2AKR1B1
SCHEMBL2269382 0.88 PTGDR2 (0.81) PTGDR2
SCHEMBL1466115 0.85 PTGDR2 (0.84) PTGDR2
SCHEMBL1785678 0.84 PTGDR2 (0.74) PTGDR2AKR1B1
SCHEMBL1782651 0.84 PTGDR2 (0.66) PTGDR2
SCHEMBL1783187 0.84 PTGDR2 (0.88) PTGDR2
SCHEMBL1784633 0.84 PTGDR2 (0.63) PTGDR2
SCHEMBL1785449 0.83 PTGDR2 (0.68) PTGDR2
SCHEMBL1786293 0.83 PTGDR2 (0.74) PTGDR2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8268878-B2 Compounds having CRTH2 antagonist activity OXAGEN LIMITED (GB) 2012-09-18 US disclosed
EP-2492268-A1 Compounds having CRTH2 antagonist activity Oxagen Limited (GB) 2012-08-29 EP disclosed
EP-2046740-B1 COMPOUNDS HAVING CRTH2 ANTAGONIST ACTIVITY OXAGEN LTD (GB) 2012-05-23 EP disclosed
US-20110268693-A1 Compounds Having CRTH2 Antagonist Activity OXAGEN LIMITED (GB) 2011-11-03 US disclosed
US-7999119-B2 Compounds having CRTH2 antagonist activity OXAGEN LIMITED (GB) 2011-08-16 US disclosed
US-20100035956-A1 Compounds Having CRTH2 Antagonist Activity OXAGEN LIMITED (GB) 2010-02-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110268693-A1 Compounds Having CRTH2 Antagonist Activity HRH2, HRH1, HRH4 PTGDR2 122/4885AKR1B1 343/4885
US-20100035956-A1 Compounds Having CRTH2 Antagonist Activity HRH2, HRH1, HRH4 PTGDR2 122/4885AKR1B1 343/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.