SCHEMBL22720222

SCHEMBL22720222

Cc1c(Br)nc(OC[C@@H]2CCCN2C)nc1N1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KRAS P01116 3/20 0.48
CHRNB2 P17787 6/20 0.42
CHRNA4 P43681 6/20 0.42
CHRNB4 P30926 4/20 0.40
CHRNA3 P32297 4/20 0.40
CHRNB1 P11230 3/20 0.40
CHRNB3 Q05901 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720224 1.00 KRAS (0.48) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22724624 0.87 KRAS (0.47) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22720351 0.83 KRAS (0.44) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22720353 0.83 KRAS (0.44) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22720294 0.81 KRAS (0.56) KRAS
SCHEMBL22720296 0.81 KRAS (0.56) KRAS
SCHEMBL19636829 0.80 KRAS (0.46) KRAS
SCHEMBL30189208 0.80 KRAS (0.46) KRAS
SCHEMBL21722205 0.79 KRAS (0.47) KRAS
SCHEMBL30834528 0.79 KRAS (0.47) KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-B Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-06-18 CN disclosed
CN-113396147-A Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-14 CN disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed