SCHEMBL22720385

SCHEMBL22720385

COC(=O)c1ncc2c(n1)CNCC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 13/20 0.46
CHRM3 P20309 2/20 0.39
HTR2B P41595 9/20 0.36
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
HTR2A P28223 1/20 0.35
HTR3A P46098 1/20 0.35
HTR6 P50406 1/20 0.35
MAPK1 P28482 1/20 0.34
CCNT1 O60563 1/20 0.33
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CCNB1 P14635 1/20 0.33
CCND1 P24385 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
CCNH P51946 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26056504 0.89 POLB (0.43) HTR2CCHRM3HTR2BCHRM4CHRM5
Hydrochloric Acid SCHEMBL28417068 0.85 CHRM3 (0.37) HTR2CCHRM3MAPK1CCNT1CDK1
SCHEMBL30648724 0.76 CDK2 (0.58) HTR2CCCNT1CDK1CDK4CCNB1
SCHEMBL26640933 0.76 CDK2 (0.58) HTR2CCCNT1CDK1CDK4CCNB1
SCHEMBL720335 0.75 CHRM3 (0.40) HTR2CCHRM3MAPK1
Hydrochloric Acid SCHEMBL22981558 0.74 CHRM3 (0.39) HTR2CCHRM3MAPK1
SCHEMBL722849 0.74 MAPK1 (0.41) HTR2CCHRM3MAPK1
SCHEMBL28949544 0.74 HTR2C (0.51) HTR2CCHRM3HTR2BCHRM4CHRM5
Trifluoroacetic Acid SCHEMBL31597693 0.74 HTR2C (0.43) HTR2CCHRM3HTR2BCHRM4CHRM5
Hydrochloric Acid SCHEMBL719328 0.73 MAPK1 (0.40) HTR2CCHRM3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239077-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE REGULATOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed