SCHEMBL22720503

SCHEMBL22720503

COC(=O)c1nc2c(c(N3CCN(C(=O)OCc4ccccc4)C(CC#N)C3)n1)CCNC2

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.41
KRAS P01116 17/20 0.38
VHL P40337 1/20 0.35
CDK7 P50613 1/20 0.35
CCNH P51946 1/20 0.35
MNAT1 P51948 1/20 0.35
SOS1 Q07889 1/20 0.35
SLC29A1 Q99808 1/20 0.34
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720500 1.00 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL28645444 0.93 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL28645449 0.93 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL19636886 0.88 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL19617263 0.88 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL29888410 0.87 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL28500547 0.87 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL19948383 0.87 IDH1 (0.41) IDH1KRASVHLCDK7CCNH
SCHEMBL30188801 0.85 IDH1 (0.40) IDH1KRASVHLCDK7CCNH
SCHEMBL26865857 0.85 IDH1 (0.40) IDH1KRASVHLCDK7CCNH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118745176-A Nitrogen-containing heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-10-08 CN disclosed
CN-118745177-A Nitrogen-containing heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-10-08 CN disclosed
CN-113423703-B Nitrogen-containing heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-08-02 CN disclosed
CN-113423703-A Nitrogen-containing heterocyclic derivative regulator, and preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-21 CN disclosed
WO-2020239077-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE REGULATOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed