SCHEMBL22720893

SCHEMBL22720893

c1ccc(Oc2ccc(-c3ccn(C4CCN(CC5CCN(C6CNC6)CC5)CC4)n3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.37
MMP9 P14780 2/20 0.37
SCN4A P35499 1/20 0.36
TNK2 Q07912 2/20 0.35
BTK Q06187 4/20 0.35
KDM2B Q8NHM5 3/20 0.34
APP P05067 1/20 0.34
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720878 0.90 SCN4A (0.42) SCN4ATNK2BTK
SCHEMBL22720927 0.87 SCN4A (0.40) SCN4ATNK2BTK
SCHEMBL28643229 0.84 PLAUR (0.37) MMP2MMP9SCN4ATNK2BTK
SCHEMBL5805292 0.81 PLAUR (0.42) SCN4ATNK2BTK
SCHEMBL27577918 0.81 SCN4A (0.49) SCN4ATNK2BTK
SCHEMBL5803668 0.78 DRD4 (0.54) SCN4A
SCHEMBL6640044 0.78 BTK (0.46) SCN4ATNK2BTKKDM2B
SCHEMBL22721138 0.78 PLAUR (0.40) SCN4ATNK2BTK
SCHEMBL22720731 0.78 SCN4A (0.40) SCN4ATNK2BTK
SCHEMBL5804770 0.77 LCK (0.47) SCN4ATNK2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118027041-A BTK inhibitor ring derivative and preparation method and pharmaceutical application thereof 西藏海思科制药有限公司 2024-05-14 CN disclosed
CN-113544130-B BTK inhibitor ring derivative and preparation method and pharmaceutical application thereof 西藏海思科制药有限公司 2024-01-09 CN disclosed
CN-113544130-A BTK inhibitor ring derivative, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2021-10-22 CN disclosed
WO-2020239103-A1 BTK INHIBITOR RING DERIVATIVE, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL APPLICATION THEREOF 四川海思科制药有限公司 2020-12-03 WO disclosed