SCHEMBL22774907

SCHEMBL22774907

COc1ccc(-c2n[nH]c(-c3ccccc3)c2CCC(=O)NO)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 5/20 0.45
CCNE1 P24864 5/20 0.45
CDK2 P24941 5/20 0.45
CDK4 P11802 4/20 0.45
CCND1 P24385 4/20 0.45
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
KMT2A Q03164 2/20 0.44
GAPDH P04406 1/20 0.44
MMP3 P08254 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
GFER P55789 1/20 0.44
HDAC1 Q13547 5/20 0.43
HDAC2 Q92769 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22769603 0.89 HDAC2 (0.47) KDM4EMMP3ALDH1A1GAAHPGD
SCHEMBL22774995 0.89 HDAC1 (0.49) CDK2MAPTGAAHDAC1HDAC2
SCHEMBL22784037 0.89 CCNE2 (0.46) CCNE2CCNE1CDK2CDK4CCND1
SCHEMBL25143291 0.85 HDAC2 (0.44) KDM4EMMP3ALDH1A1GAAHPGD
SCHEMBL22769610 0.82 HDAC1 (0.50) KDM4EALDH1A1GAAHPGDHDAC1
SCHEMBL22774997 0.78 HDAC1 (0.46) CDK2KDM4EMAPTKMT2AMEN1
SCHEMBL22769602 0.77 KDM4E (0.45) CCNE2CCNE1CDK2CDK4CCND1
SCHEMBL17279858 0.75 TSHR (0.43) CCNE2CCNE1CDK2CDK4CCND1
SCHEMBL1128878 0.75 CA1 (0.47) CDK2KDM4EMAPTALDH1A1GAA
SCHEMBL25143532 0.75 PDE4A (0.48) KDM4EMAPTKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3986868-A1 HETEROAROMATIC INHIBITORS OF ASTACIN PROTEINASES Vivoryon Therapeutics N.V. (DE) 2022-04-27 EP disclosed
WO-2020249760-A1 HETEROAROMATIC INHIBITORS OF ASTACIN PROTEINASES VIVORYON THERAPEUTICS AG (DE) 2020-12-17 WO disclosed