SCHEMBL22807447

SCHEMBL22807447

C=CC(=O)Nc1c(F)cccc1Nc1nc(Cl)ncc1Cl

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK3 P27361 15/20 0.52
EGFR P00533 2/20 0.48
BTK Q06187 2/20 0.48
MAPK1 P28482 2/20 0.48
MAP2K1 Q02750 1/20 0.48
FGFR4 P22455 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29549982 1.00 MAPK3 (0.52) MAPK3EGFRBTKMAPK1MAP2K1
SCHEMBL602415 0.85 MAPK3 (0.40) MAPK3EGFR
SCHEMBL15938232 0.83 MAPK3 (0.66) MAPK3EGFRMAPK1MAP2K1
SCHEMBL29251292 0.80 EGFR (0.55) MAPK3EGFRBTK
SCHEMBL30366835 0.80 FGFR4 (0.56) MAPK3MAPK1MAP2K1FGFR4
SCHEMBL30584603 0.80 EGFR (0.55) MAPK3EGFRBTK
SCHEMBL16370812 0.79 MAPK3 (0.55) MAPK3EGFRMAPK1MAP2K1
SCHEMBL29549741 0.79 MAPK3 (0.70) MAPK3BTK
SCHEMBL15938675 0.79 MAPK3 (0.70) MAPK3BTK
SCHEMBL22807504 0.78 MAP3K7 (0.79) EGFRBTKMAPK1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12365664-B2 Small molecule inhibitors of SRC tyrosine kinase DANA-FARBER CANCER INSTITUTE, INC. (US) 2025-07-22 US disclosed
US-20220267294-A1 SMALL MOLECULE INHIBITORS OF SRC TYROSINE KINASE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2022-08-25 US disclosed
EP-3986411-A1 SMALL MOLECULE INHIBITORS OF SRC TYROSINE KINASE Dana-Farber Cancer Institute, Inc. (US) 2022-04-27 EP disclosed
WO-2020257385-A1 SMALL MOLECULE INHIBITORS OF SRC TYROSINE KINASE DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-12-24 WO disclosed
WO-2020257385-A1 SMALL MOLECULE INHIBITORS OF SRC TYROSINE KINASE DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12365664-B2 Small molecule inhibitors of SRC tyrosine kinase SRC, CTTN, LCK MAPK3 273/4885EGFR 127/4885BTK 8/4885
US-20220267294-A1 SMALL MOLECULE INHIBITORS OF SRC TYROSINE KINASE SRC, CTTN, LCK MAPK3 273/4885EGFR 127/4885BTK 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.