SCHEMBL22809485

SCHEMBL22809485

C[C@@H](N)COc1ncc(C(F)(F)I)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 2/20 0.37
KMT2A Q03164 1/20 0.37
HPGD P15428 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809581 0.89 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL3649246 0.89 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C19SMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL28350721 0.87 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL19075622 0.72 SCN9A (0.43) CYP1A2CYP3A4CYP2C19
SCHEMBL28354400 0.70 SMN1; SMN2 (0.49) CYP1A2CYP3A4CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL19083934 0.70 SCN9A (0.41) CYP3A4CYP2C19
SCHEMBL14051590 0.68 CYP1A2 (0.55) CYP1A2CYP3A4CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL20697770 0.68 SCN9A (0.40) CYP1A2CYP3A4CYP2C19
SCHEMBL22809491 0.68 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL22809492 0.68 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed