SCHEMBL22828751

SCHEMBL22828751

Cc1ccncc1-c1ncccc1C

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.59
CYP11B1 P15538 4/20 0.50
CYP11B2 P19099 4/20 0.50
METAP2 P50579 1/20 0.46
GPBAR1 Q8TDU6 1/20 0.42
CYP17A1 P05093 7/20 0.41
CYP1A2 P05177 5/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
PDE10A Q9Y233 1/20 0.40
WNT1 P04628 1/20 0.40
PTGS2 P35354 1/20 0.40
NPY5R Q15761 1/20 0.40
ABL1 P00519 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30546874 0.84 CYP2A6 (0.46) CYP2A6CYP11B1CYP11B2CYP17A1CYP1A2
SCHEMBL16149264 0.84 CYP2A6 (0.46) CYP2A6CYP11B1CYP11B2GPBAR1CYP17A1
SCHEMBL15778479 0.80 CYP2A6 (0.54) CYP2A6METAP2GPBAR1NOS3NOS1
SCHEMBL30442955 0.80 CYP2A6 (0.54) CYP2A6METAP2GPBAR1NOS3NOS1
SCHEMBL4160810 0.79 CYP2A6 (0.52) CYP2A6METAP2CYP1A2NOS3NOS1
SCHEMBL15243551 0.78 CYP17A1 (0.44) CYP2A6CYP11B1CYP11B2CYP17A1CYP1A2
SCHEMBL12097338 0.78 CYP2A6 (0.51) CYP2A6METAP2GPBAR1CYP1A2NOS3
SCHEMBL18174651 0.77 CYP2A6 (0.51) CYP2A6CYP11B1CYP11B2CYP17A1CYP1A2
SCHEMBL196235 0.76 CYP2A6 (0.61) CYP2A6METAP2NOS3NOS1NOS2
SCHEMBL31252534 0.76 CYP2A6 (0.61) CYP2A6METAP2NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020253458-A1 CDK KINASE INHIBITOR 北京睿熙生物科技有限公司 2020-12-24 WO disclosed