SCHEMBL22832997

SCHEMBL22832997

Cn1cnnc1C1(c2cccc(Br)c2)CC2(CC2)C1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CBLB Q13191 19/20 0.41
CBL P22681 15/20 0.41
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
CBLC Q9ULV8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25179648 0.95 CBLB (0.44) CBLBCBLCTSDBACE1
SCHEMBL30374080 0.95 CBLB (0.44) CBLBCBLCTSDBACE1
SCHEMBL30521214 0.89 CBLB (0.46) CBLBCBL
SCHEMBL30373880 0.89 CBLB (0.38) CBLBCBLCBLC
SCHEMBL25183728 0.89 CBLB (0.38) CBLBCBLCBLC
SCHEMBL30374453 0.89 CBLB (0.40) CBLBCBLCBLC
SCHEMBL32686461 0.89 CBLB (0.40) CBLBCBLCBLC
SCHEMBL25183642 0.89 CBLB (0.40) CBLBCBLCBLC
SCHEMBL24662646 0.88 CBLB (0.41) CBLBCBLCTSDBACE1CBLC
SCHEMBL30374240 0.88 CBLB (0.41) CBLBCBLCTSDBACE1CBLC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260028336-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2026-01-29 US disclosed
EP-4653436-A1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND USE THEREOF GUANGZHOU YUFAN NANTU BIOTECHNOLOGIES CO., LTD (CN) 2025-11-26 EP disclosed
CN-114364670-B Substituted benzyl-triazole compound for Cbl-b inhibition and further application thereof 纽力克斯治疗公司 2025-06-13 CN disclosed
EP-4558501-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF Arcus Biosciences, Inc. (US) 2025-05-28 EP disclosed
US-20250136590-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. 2025-05-01 US disclosed
US-12234230-B2 Substituted benzyl-triazole compounds for Cbl-b inhibition, and further uses thereof NURIX THERAPEUTICS, INC. (US) 2025-02-25 US disclosed
WO-2024153240-A1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND USE THEREOF 珠海宇繁生物科技有限责任公司 2024-07-25 WO disclosed
WO-2024105563-A1 SUBSTITUTED BICYCLIC PYRIDONE DERIVATIVES PFIZER INC. (US) 2024-05-23 WO disclosed
WO-2024020034-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2024-01-25 WO disclosed
WO-2024020034-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2024-01-25 WO disclosed
US-20230150991-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. 2023-05-18 US disclosed
US-20230150991-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. 2023-05-18 US disclosed
US-20230150991-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. 2023-05-18 US disclosed
US-11401267-B2 Substituted benzyl-triazole compounds for Cbl-b inhibition, and further uses thereof NURIX THERAPEUTICS, INC. (US) 2022-08-02 US disclosed
EP-3990117-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF Nurix Therapeutics, Inc. (US) 2022-05-04 EP disclosed
CN-114364670-A Substituted benzyl-triazoles for Cbl-b inhibition and further uses thereof 纽力克斯治疗公司 2022-04-15 CN disclosed
US-20210053961-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. 2021-02-25 US disclosed
US-20210053961-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. 2021-02-25 US disclosed
WO-2020264398-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. (US) 2020-12-30 WO disclosed
WO-2020264398-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF NURIX THERAPEUTICS, INC. (US) 2020-12-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11401267-B2 Substituted benzyl-triazole compounds for Cbl-b inhibition, and further uses thereof CBL, CBLB, CBLC CBLB 2/4885CBL 1/4885CTSD 1404/4885
US-20230150991-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF CBL, CBLB, CBLC CBLB 2/4885CBL 1/4885CTSD 1404/4885
US-20260028336-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF CBLB, CBL, CBLC CBLB 1/4885CBL 2/4885CTSD 4391/4885
US-12234230-B2 Substituted benzyl-triazole compounds for Cbl-b inhibition, and further uses thereof CBL, CBLB, CBLC CBLB 2/4885CBL 1/4885CTSD 1404/4885
US-20250136590-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF CBL, CBLB, CBLC CBLB 2/4885CBL 1/4885CTSD 1404/4885
US-20210053961-A1 SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FURTHER USES THEREOF CBL, CBLB, CBLC CBLB 2/4885CBL 1/4885CTSD 1404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.