SCHEMBL2283457

SCHEMBL2283457

CC(C)(C)C#Cc1cc(N(C(=O)[C@H]2CC[C@H](C)CC2)[C@H]2CCN(C(=O)OC3CCCNC3)C2)c(C(=O)O)s1

nearest known ligand 0.56

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.56
CYP2E1 P05181 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12439631 1.00 NR1I2 (0.56) NR1I2CYP2E1
SCHEMBL2218884 1.00 NR1I2 (0.56) NR1I2CYP2E1
SCHEMBL2216739 0.96 NR1I2 (0.57) NR1I2CYP2E1
SCHEMBL12439473 0.93 NR1I2 (0.60) NR1I2CYP2E1
SCHEMBL2219255 0.92 NR1I2 (0.56) NR1I2CYP2E1
SCHEMBL12439447 0.92 NR1I2 (0.60) NR1I2CYP2E1
SCHEMBL12514090 0.90 NR1I2 (0.42) NR1I2CYP2E1
SCHEMBL12439472 0.88 NR1I2 (0.62) NR1I2CYP2E1
SCHEMBL12439627 0.88 NR1I2 (0.55) NR1I2CYP2E1
SCHEMBL12439624 0.88 NR1I2 (0.55) NR1I2CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523951-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES Gilead Sciences, Inc. (US) 2012-11-21 EP disclosed
WO-2011088303-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES , INC. (US) 2011-07-21 WO disclosed