SCHEMBL22838686

SCHEMBL22838686

CNC(=O)c1c(F)cnc2c(CCNc3cc(-c4ccc(OCC5CC5)nc4)ncn3)cccc12

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.36
WDR5 P61964 2/20 0.34
USP2 O75604 5/20 0.34
CYP1A2 P05177 5/20 0.34
CYP3A4 P08684 5/20 0.34
CLK4 Q9HAZ1 5/20 0.34
CYP2C19 P33261 4/20 0.34
CYP2D6 P10635 4/20 0.34
ALDH1A1 P00352 3/20 0.34
ALOX15 P16050 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP2C9 P11712 1/20 0.34
SYK P43405 1/20 0.34
HSD17B10 Q99714 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33
ACACB O00763 3/20 0.33
ACACA Q13085 2/20 0.33
GABRA5 P31644 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22838575 0.90 GCK (0.40) PTGESUSP2CYP1A2CYP3A4CLK4
SCHEMBL19355619 0.89 CYP1A2 (0.40) USP2CYP1A2CYP3A4CLK4CYP2C19
SCHEMBL19355604 0.88 FFAR4 (0.37) USP2CYP1A2CYP3A4CLK4CYP2C19
SCHEMBL19905428 0.87 CYP1A2 (0.38) PTGESWDR5USP2CYP1A2CYP3A4
SCHEMBL19905429 0.86 CYP1A2 (0.35) USP2CYP1A2CYP3A4CLK4CYP2C19
SCHEMBL19905405 0.86 FEN1 (0.36) USP2CYP1A2CYP3A4CLK4CYP2C19
SCHEMBL19355618 0.86 CYP1A2 (0.37) USP2CYP1A2CYP3A4CLK4CYP2C19
SCHEMBL17634848 0.85 PRKDC (0.42) PTGESWDR5SYKACACBACACA
SCHEMBL19905266 0.84 PRKDC (0.37) USP2CYP1A2CYP3A4CLK4CYP2C19
SCHEMBL19905175 0.84 CYP1A2 (0.40) USP2CYP1A2CYP3A4CLK4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3459942-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2020-12-30 EP disclosed