SCHEMBL22853005

SCHEMBL22853005

Cc1cc(F)ccc1Nc1cc(C(F)F)c(F)cc1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY4 P51582 1/20 0.46
IDO1 P14902 2/20 0.43
CLCN2 P51788 1/20 0.43
DHODH Q02127 5/20 0.41
MKNK2 Q9HBH9 1/20 0.41
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
FABP3 P05413 1/20 0.40
FABP4 P15090 1/20 0.40
MAP2K1 Q02750 2/20 0.39
FTO Q9C0B1 1/20 0.39
MAP2K2 P36507 1/20 0.39
MPO P05164 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294522 1.00 P2RY4 (0.46) P2RY4IDO1CLCN2DHODHMKNK2
SCHEMBL30294815 0.89 CLCN2 (0.49) P2RY4IDO1CLCN2DHODHMKNK2
SCHEMBL22853350 0.89 CLCN2 (0.49) P2RY4IDO1CLCN2DHODHMKNK2
SCHEMBL22853121 0.88 IDO1 (0.48) P2RY4IDO1CLCN2DHODHMKNK2
SCHEMBL30294377 0.88 IDO1 (0.48) P2RY4IDO1CLCN2DHODHMKNK2
SCHEMBL22853048 0.87 MAPK13 (0.39) MAPK13MAPK12MAPK11MAPK14ALDH1A1
SCHEMBL30294637 0.87 MAPK13 (0.39) MAPK13MAPK12MAPK11MAPK14ALDH1A1
SCHEMBL22853346 0.86 IDO1 (0.50) P2RY4IDO1CLCN2DHODHMKNK2
SCHEMBL30294440 0.86 IDO1 (0.50) P2RY4IDO1CLCN2DHODHMKNK2
SCHEMBL22853383 0.83 P2RY4 (0.56) P2RY4IDO1CLCN2DHODHMKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020261114-A1 2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-12-30 WO disclosed