SCHEMBL22853045

SCHEMBL22853045

CCOC(=O)c1ccc(C)cc1Nc1ccc(F)cc1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K2 P36507 1/20 0.43
MAP2K1 Q02750 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
POLB P06746 1/20 0.43
KDM4E B2RXH2 3/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CDC25B P30305 3/20 0.42
TSHR P16473 1/20 0.42
MRGPRX1 Q96LB2 1/20 0.41
CDC25A P30304 1/20 0.39
CDC25C P30307 1/20 0.39
NPSR1 Q6W5P4 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294599 1.00 MAP2K2 (0.43) MAP2K2MAP2K1SMN1; SMN2TDP1POLB
SCHEMBL22853359 0.87 KDM4E (0.42) MAP2K2MAP2K1SMN1; SMN2TDP1POLB
SCHEMBL30294715 0.87 KDM4E (0.42) MAP2K2MAP2K1SMN1; SMN2TDP1POLB
SCHEMBL30294254 0.84 CLCN2 (0.46)
SCHEMBL22853007 0.84 CLCN2 (0.46)
SCHEMBL22853027 0.81 RECQL (0.42) SMN1; SMN2POLBKDM4ELMNACYP1A2
SCHEMBL30294633 0.81 RECQL (0.42) SMN1; SMN2POLBKDM4ELMNACYP1A2
SCHEMBL22853053 0.81 MRGPRX4 (0.42) SMN1; SMN2TDP1POLBKDM4ELMNA
SCHEMBL30294656 0.81 MRGPRX4 (0.42) SMN1; SMN2TDP1POLBKDM4ELMNA
SCHEMBL24553052 0.77 MAPT (0.42) SMN1; SMN2TDP1KDM4ELMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020261114-A1 2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-12-30 WO disclosed