SCHEMBL2286133

SCHEMBL2286133

Cc1noc(C)c1-c1c(C=O)c2c(F)ccc(F)c2n1-c1ccc(O)cc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.48
BRD4 O60885 9/20 0.36
PIK3CD O00329 1/20 0.33
EDNRA P25101 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
LMNA P02545 1/20 0.31
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2288272 0.88 ERN1 (0.39) ERN1BRD4PIK3CDKMT2ALMNA
SCHEMBL2288274 0.88 ERN1 (0.39) ERN1BRD4PIK3CDKMT2ALMNA
SCHEMBL2287848 0.85 ERN1 (0.44) ERN1BRD4PIK3CDLMNA
SCHEMBL2283182 0.85 ERN1 (0.42) ERN1BRD4PIK3CDKMT2ALMNA
SCHEMBL2282817 0.82 ERN1 (0.43) ERN1BRD4PIK3CDFFAR1
SCHEMBL2312429 0.81 ERN1 (0.36) ERN1BRD4PIK3CDKMT2A
SCHEMBL2146602 0.80 ERN1 (0.45) ERN1BRD4PIK3CDLMNA
SCHEMBL2307790 0.78 ERN1 (0.34) ERN1BRD4PIK3CDKMT2ALMNA
SCHEMBL2307797 0.78 ERN1 (0.34) ERN1BRD4PIK3CD
SCHEMBL2312965 0.78 ERN1 (0.34) ERN1BRD4PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110201555-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-08-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110201555-A1 NOVEL ESTROGEN RECEPTOR LIGANDS ESR1, ESRRA, GPER1 ERN1 384/4885BRD4 891/4885PIK3CD 4139/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.