SCHEMBL22878645

SCHEMBL22878645

CC(N=O)c1cc(=O)c(O)cn1-c1cccc(-c2cncc3ccccc23)c1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
COMT P21964 9/20 0.53
NTSR1 P30989 2/20 0.40
CYP11B1 P15538 3/20 0.39
CYP11B2 P19099 3/20 0.39
ERN1 O75460 1/20 0.39
CCNC P24863 3/20 0.38
CDK8 P49336 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2433183 0.89 COMT (0.67) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL6901113 0.89 COMT (0.55) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL6899331 0.88 COMT (0.69) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL6900457 0.87 COMT (0.52) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL6901187 0.87 COMT (0.53) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL22878679 0.86 COMT (0.46) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL6901267 0.85 COMT (0.68) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL14816273 0.84 COMT (0.50) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL14815792 0.83 COMT (0.54) COMTNTSR1CYP11B1CYP11B2ERN1
SCHEMBL6901266 0.83 COMT (0.50) COMTNTSR1CYP11B1CYP11B2ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2542076-B1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME (US) 2021-01-13 EP disclosed