SCHEMBL22878680

SCHEMBL22878680

CC(O)c1cc(=O)c(O)cn1-c1cccc(-c2c(O)cnc3[nH]ccc23)c1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
COMT P21964 10/20 0.61
CDK8 P49336 1/20 0.36
PDE4A P27815 1/20 0.34
KCNH2 Q12809 1/20 0.34
JAK3 P52333 1/20 0.32
RPS6KA3 P51812 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22878726 0.93 COMT (0.59) COMTCDK8RPS6KA3
SCHEMBL2467436 0.92 COMT (0.58) COMTCDK8
SCHEMBL6901891 0.84 COMT (0.65) COMTCDK8
SCHEMBL14816251 0.82 COMT (0.60) COMT
SCHEMBL14815722 0.81 COMT (0.44) COMT
SCHEMBL14816399 0.79 COMT (0.44) COMTRPS6KA3
SCHEMBL14816287 0.79 COMT (0.66) COMTCDK8
SCHEMBL6899372 0.79 COMT (0.44) COMT
SCHEMBL2439128 0.77 COMT (1.00) COMT
SCHEMBL2433208 0.76 COMT (0.41) COMTJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2542076-B1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME (US) 2021-01-13 EP disclosed