SCHEMBL2288995

SCHEMBL2288995

CCOC(=O)c1cccc(N2C[C@@H]3CCCN3c3nc(SC)ncc3C2=O)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 12/20 0.52
CACNA2D2 Q9NY47 1/20 0.52
SLC6A2 P23975 8/20 0.49
BTK Q06187 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.42
ALOX5 P09917 1/20 0.40
MAPT P10636 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2288362 1.00 CACNA2D1 (0.52) CACNA2D1CACNA2D2SLC6A2BTKMEN1
SCHEMBL2289695 0.88 CACNA2D1 (0.51) CACNA2D1CACNA2D2SLC6A2MEN1KMT2A
SCHEMBL2289702 0.88 CACNA2D1 (0.51) CACNA2D1CACNA2D2SLC6A2MEN1KMT2A
SCHEMBL2288797 0.87 CACNA2D1 (0.52) CACNA2D1CACNA2D2SLC6A2
SCHEMBL2288791 0.87 CACNA2D1 (0.52) CACNA2D1CACNA2D2SLC6A2
SCHEMBL2293095 0.87 CACNA2D1 (0.70) CACNA2D1CACNA2D2SLC6A2
SCHEMBL2292019 0.86 CACNA2D1 (0.51) CACNA2D1CACNA2D2SLC6A2MEN1KMT2A
SCHEMBL2292026 0.86 CACNA2D1 (0.51) CACNA2D1CACNA2D2SLC6A2MEN1KMT2A
SCHEMBL2289722 0.84 CACNA2D1 (0.48) CACNA2D1CACNA2D2SLC6A2
SCHEMBL2289725 0.84 CACNA2D1 (0.48) CACNA2D1CACNA2D2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998954-B2 Pyrimidodiazepinone derivative KYOWA HAKKO KIRIN CO., LTD. (JP) 2011-08-16 US disclosed