SCHEMBL22901583

SCHEMBL22901583

COc1cccc(COc2cccc3ccc(-c4nc(C)cc(C)n4)nc23)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
HTT P42858 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
ABCB1 P08183 6/20 0.47
HTR1A P08908 3/20 0.47
DRD2 P14416 2/20 0.47
GCK P35557 1/20 0.46
FFAR1 O14842 1/20 0.44
MAOB P27338 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
SGMS2 Q8NHU3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22901547 0.90 MEN1 (0.51) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901571 0.90 MAPT (0.48) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901567 0.88 MAPT (0.51) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901578 0.88 MAOB (0.48) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901554 0.88 MAPT (0.51) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901562 0.87 MAPT (0.50) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL9951098 0.86 MEN1 (0.67) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901575 0.85 MAPT (0.48) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901572 0.84 MEN1 (0.48) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL22901560 0.84 MAPT (0.47) MAPTHTTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021008588-A1 CLASS OF PYRIMIDINE QUINOLINE DERIVATIVES AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 广州新民培林医药科技有限公司 2021-01-21 WO disclosed