SCHEMBL22904753

SCHEMBL22904753

CC(C)(C)OC(=O)N1CC2(CC2)C[C@H]1c1nc(I)c2c(Cl)nccn12

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 14/20 0.41
TNK2 Q07912 1/20 0.35
POLB P06746 1/20 0.33
KCNK3 O14649 2/20 0.31
KCNK9 Q9NPC2 2/20 0.31
NAMPT P43490 1/20 0.31
EIF2AK4 Q9P2K8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21461728 0.89 BTK (0.41) BTKTNK2POLBKCNK3KCNK9
SCHEMBL22904751 0.89 BTK (0.50) BTKTNK2
SCHEMBL20415500 0.82 BTK (0.36) BTKTNK2POLBKCNK3KCNK9
SCHEMBL21461736 0.82 BTK (0.36) BTKTNK2POLBKCNK3KCNK9
SCHEMBL30565868 0.81 BTK (0.42) BTKPOLB
SCHEMBL20415459 0.80 BTK (0.50) BTKTNK2
SCHEMBL20415461 0.80 BTK (0.50) BTKTNK2
SCHEMBL26791467 0.75 TNK2 (0.38) BTKTNK2POLBKCNK3KCNK9
SCHEMBL26791423 0.74 TNK2 (0.50) BTKTNK2POLB
SCHEMBL20415501 0.74 BTK (0.36) BTKNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113993871-B BTK inhibitors containing 5-azacycloheptane 正大天晴药业集团股份有限公司 2023-08-01 CN disclosed
WO-2021008441-A1 BTK INHIBITOR CONTAINING 5-AZASPIROHEPTANE 正大天晴药业集团股份有限公司 2021-01-21 WO disclosed