SCHEMBL22909488

SCHEMBL22909488

COc1ccc(C2=NN(c3ccccn3)C(=O)C2)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 12/20 1.00
PDCD1 Q15116 10/20 1.00
PDE4B Q07343 6/20 0.56
PDE4A P27815 5/20 0.56
PDE4C Q08493 5/20 0.56
PDE4D Q08499 5/20 0.56
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22908681 0.84 CD274 (1.00) CD274PDCD1GAAL3MBTL1KDM4E
SCHEMBL15521537 0.83 CD274 (0.76) CD274PDCD1ALDH1A1GAA
SCHEMBL15058050 0.83 PDE4B (0.79) CD274PDCD1PDE4BPDE4APDE4C
SCHEMBL22908675 0.81 CD274 (1.00) CD274PDCD1ALDH1A1GAAHPGD
SCHEMBL22908607 0.79 CD274 (1.00) CD274PDCD1GAAL3MBTL1KDM4E
SCHEMBL16979677 0.79 CD274 (0.74) CD274PDCD1ALDH1A1GAAHPGD
SCHEMBL22909491 0.79 CD274 (1.00) CD274PDCD1ALDH1A1GAAKDM4E
SCHEMBL22908621 0.77 CD274 (1.00) CD274PDCD1GAAL3MBTL1KDM4E
SCHEMBL15057911 0.75 PDCD1 (0.60) CD274PDCD1PDE4BPDE4APDE4C
SCHEMBL28265426 0.75 PDE4B (0.60) CD274PDCD1PDE4BPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021009384-A1 NOVEL PYRAZOLONE DERIVATIVES AS PD-1/PD-L1 INTERACTION INHIBITORS CENTRE HOSPITALIER REGIONAL UNIVERSITAIRE DE LILLE (FR) 2021-01-21 WO disclosed