SCHEMBL22926535

SCHEMBL22926535

COc1cc(N2CCOC[C@H]2C)nc(Nc2cc[nH]n2)c1C=N

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ATR Q13535 19/20 0.47
ATRIP Q8WXE1 16/20 0.45
CHEK1 O14757 3/20 0.40
PDCD1 Q15116 3/20 0.40
CD274 Q9NZQ7 3/20 0.40
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24708105 0.87 ATR (0.43) ATRATRIPCHEK1PDCD1CD274
SCHEMBL22926536 0.85 ATR (0.46) ATRATRIPCHEK1PDCD1CD274
SCHEMBL22926602 0.85 ATR (0.46) ATRATRIPCHEK1PDCD1CD274
SCHEMBL24708215 0.84 ATR (0.46) ATRATRIPCHEK1PDCD1CD274
SCHEMBL22926606 0.83 ATR (0.38) ATRATRIPCHEK1PDCD1CD274
SCHEMBL22926485 0.83 ATR (0.46) ATRATRIP
SCHEMBL22926760 0.83 ATR (0.46) ATRATRIPCHEK1PDCD1CD274
SCHEMBL24694801 0.82 ATR (0.37) ATRATRIPCHEK1PDCD1CD274
SCHEMBL23514856 0.82 ATR (0.41) ATRATRIPCHEK1PDCD1CD274
SCHEMBL24695084 0.82 ATR (0.37) ATRATRIPCHEK1PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021012049-A1 SUBSTITUTED 2-MORPHOLINOPYRIDINE DERIVATIVES AS ATR KINASE INHIBITORS REPARE THERAPEUTICS INC. (CA) 2021-01-28 WO disclosed