SCHEMBL22927451

SCHEMBL22927451

COc1ccc2c(c1)C(=O)N(C)C(=O)C2(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
KDM4E B2RXH2 2/20 0.60
ALOX15 P16050 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
PGR P06401 1/20 0.49
APAF1 O14727 1/20 0.44
MAPT P10636 1/20 0.44
APP P05067 1/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
POLB P06746 2/20 0.41
ADAM17 P78536 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
PDE3A Q14432 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22917698 0.82 KDM4E (0.57) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL3050512 0.81 MEN1 (0.51) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL11747568 0.80 TDP1 (0.70) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL11741086 0.78 TDP1 (0.67) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL26930617 0.78 TDP1 (0.63) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL11738163 0.78 TDP1 (0.63) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL7650360 0.78 NR1H2 (0.43) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL28250120 0.78 MAPT (0.60) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL11735674 0.77 TDP1 (0.62) ALDH1A1KDM4EALOX15TDP1MEN1
SCHEMBL21586561 0.76 TDP1 (0.63) ALDH1A1KDM4EALOX15TDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021015841-A1 BORON-CONTAINING PHARMACOPHORE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2021-01-28 WO disclosed