SCHEMBL22927645

SCHEMBL22927645

N#Cc1cccc(C(N)c2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
GRM4 Q14833 1/20 0.45
TNF P01375 1/20 0.43
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HPGDS O60760 1/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 1/20 0.41
ENPP2 Q13822 1/20 0.40
KIF11 P52732 1/20 0.40
KCNA5 P22460 1/20 0.39
GSK3B P49841 1/20 0.39
TACR1 P25103 1/20 0.39
MRGPRX1 Q96LB2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29434770 1.00 TSHR (0.48) TSHRGRM4TNFSLC6A2SLC6A4
Hydrochloric Acid SCHEMBL29908241 0.98 TSHR (0.46) TSHRGRM4TNFSLC6A2SLC6A4
SCHEMBL1528610 0.86 CNR1 (0.44)
SCHEMBL1528612 0.86 CNR1 (0.44)
Hydrochloric Acid SCHEMBL1500635 0.84 CNR1 (0.43)
Hydrochloric Acid SCHEMBL1500633 0.84 CNR1 (0.43)
SCHEMBL2939744 0.82 GRM4 (0.44) TSHRGRM4TNFSLC6A2SLC6A4
SCHEMBL2982599 0.82 TSHR (0.54) TSHR
SCHEMBL17196263 0.81 KDM4E (0.40) TSHRGRM4TNFSLC6A2SLC6A4
SCHEMBL2324270 0.81 DPP4 (0.38) GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114174290-A Modulators of TREX1 星座制药公司 2022-03-11 CN disclosed
WO-2021016317-A1 MODULATORS OF TREX1 CONSTELLATION PHARMACEUTICALS, INC. (US) 2021-01-28 WO disclosed