SCHEMBL22940779

SCHEMBL22940779

Cc1cccc(-c2ccc[nH]2)n1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.58
CCR8 P51685 1/20 0.58
METAP2 P50579 1/20 0.46
CYP2A6 P11509 1/20 0.42
TGFBR1 P36897 9/20 0.39
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
PARP1 P09874 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C8 P10632 1/20 0.38
KDM4C Q9H3R0 1/20 0.37
MAPK14 Q16539 1/20 0.36
ADORA2A P29274 1/20 0.35
PDGFRB P09619 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20019709 0.85 PARP1 (0.44) CCR1CCR8PARP1KDM4CADORA2A
SCHEMBL13831067 0.85 CCR1 (0.41) CCR1CCR8METAP2CYP2A6NOS3
SCHEMBL3992598 0.83 CCR1 (0.47) CCR1CCR8METAP2CYP2A6TGFBR1
SCHEMBL310731 0.79 CCR1 (0.50) CCR1CCR8METAP2CYP2A6TGFBR1
SCHEMBL17708555 0.77 ADORA2A (0.39) CCR1CCR8NOS3NOS2PARP1
SCHEMBL3745071 0.75 CCR1 (0.62) CCR1CCR8METAP2CYP2A6TGFBR1
SCHEMBL1456972 0.75 CCR1 (0.62) CCR1CCR8METAP2CYP2A6TGFBR1
SCHEMBL196966 0.75 CCR1 (1.00) CCR1CCR8METAP2CYP2A6TGFBR1
SCHEMBL30511194 0.75 CCR1 (1.00) CCR1CCR8METAP2CYP2A6TGFBR1
SCHEMBL29388304 0.75 CCR1 (1.00) CCR1CCR8METAP2CYP2A6TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11584745-B2 Aromatic heterocyclic compound, intermediate thereof, preparation method therefor, and pharmaceutical composition and use thereof SHANGHAI YINGLI PHARMACEUTICAL CO., LTD (CN) 2023-02-21 US disclosed
US-20210032241-A1 AROMATIC HETEROCYCLIC COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF SHANGHAI YINGLI PHARMACEUTICAL CO., LTD (CN) 2021-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210032241-A1 AROMATIC HETEROCYCLIC COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF ALK, NOTUM, WEE1 CCR1 1379/4885CCR8 607/4885METAP2 2685/4885
US-11584745-B2 Aromatic heterocyclic compound, intermediate thereof, preparation method therefor, and pharmaceutical composition and use thereof ALK, NOTUM, WEE1 CCR1 1379/4885CCR8 607/4885METAP2 2685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.